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6-tetra-O-actyl-1-C-[4-chloro-3-[[4-[[(3S)-tetrahydrofu-ran-3-yl]oxy] phenyl]

6-tetra-O-actyl-1-C-[4-chloro-3-[[4-[[(3S)-tetrahydrofu-ran-3-yl]oxy] phenyl]

Sharaxaad Gaaban:

Qaaciddada molecular: C31H35ClO11
Miisaanka molecular: 619.056
CAS no: 915095-99-7


Faahfaahinta Alaabta

Tags Product

Codsiga

Alaabtani waa kiniin huruud ah oo khafiif ah oo dahaarka leh, caddaan ama ku dhawaad ​​cad ka dib markii laga saaro daahan.

Tilmaamaha
Alaabtani waxay ku habboon tahay daawaynta nooca 2aad ee sonkorowga.

monotherapy
Alaabtan waxa lala isticmaalaa xakamaynta cuntada iyo jimicsiga si loo hagaajiyo xakamaynta sonkorta dhiigga ee bukaanka qaba nooca 2 ee sonkorowga.

Waxaa loo isticmaalaa in lagu daro metformin hydrochloride
Marka metformin hydrochloride keligiis uusan si wax ku ool ah u xakameyn karin sonkorta dhiigga, badeecadan waxaa loo isticmaali karaa in lagu daro metformin hydrochloride si loo hagaajiyo xakameynta sonkorta dhiigga bukaanka qaba nooca 2 ee sonkorowga iyadoo lagu saleynayo cuntada iyo jimicsiga.

Waxaa loo isticmaalaa in lagu daro metformin hydrochloride iyo sulfonylureas.
Marka la isku daro isticmaalka metformin hydrochloride iyo sulfonylureas aysan si wax ku ool ah u xakameyn karin sonkorta dhiigga, alaabtan waxaa loo isticmaali karaa in lagu daro metformin hydrochloride iyo sulfonylureas si loo hagaajiyo xakamaynta sonkorta dhiigga ee bukaanka qaba nooca 2 ee sonkorowga iyadoo lagu saleynayo cuntada iyo jimicsiga.

Xayiraadaha daawada
Alaabtan laguma talinayo bukaanka nooca 1-aad ee sonkorowga ama daawaynta ketoacidosis-ka macaanka.

Tilmaamid
(1) 10 mg;(2) 25 mg.

Qiyaasta
Qiyaasta lagu taliyay
Qiyaasta lagu taliyey ee alaabtani waa 10 mg subaxdii, hal mar maalintii, calool madhan ama cuntada ka dib.Bukaannada u dulqaata alaabtan, qiyaasta waxaa lagu kordhin karaa 25 mg (eeg [Tijaabooyin Caafimaad]).
Bukaannada qaba hypovolemia, waxaa lagula talinayaa in la saxo hypovolemia ka hor inta aan la bilaabin isticmaalka alaabtan (eeg [Taxadirrada]).

Bukaanka qaba cillad kelyaha.
Waxaa lagu talinayaa in la qiimeeyo shaqada kelyaha ka hor inta aanad bilaabin isticmaalka alaabtan, ka dibna waa in si joogto ah loo qiimeeyaa.
Bukaannada eGFR ay ka hooseeyaan 45 ml/min/1.73 m2 waa in aanay isticmaalin alaabtan.
Bukaanka leh eGFR ka sarreeya ama la mid ah 45 mL/min/1.73 m2 uma baahna inay hagaajiyaan qiyaasta.
Haddii eGFR uu si joogto ah uga hooseeyo 45 mL/min/1.73 m2, alaabtan waa in la joojiyaa (eeg [Taxadir]).

Bukaanka qaba dhaawaca beerka.
Bukaanka qaba dhaawaca beerka uma baahna inay hagaajiyaan qiyaasta.Soo-gaadhista Enpagliflozin ayaa kor u kacday bukaannada qaba dhaawaca beerka ee daran.Waayo-aragnimada daaweynta bukaannada qaba dhaawaca beerka daran waa mid xaddidan, sidaas darteed, laguma talinayo qaybtan dadweynaha.

Heerka:heerka ganacsiga
daahirnimo≥99.0%

Dibadda:cad ilaa budo cad
Xidhmada25kg/durbaan

Khadka Alaabta isku-dhafan

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Shahaado

JIN DUN Medical ayaa lehShahaadada ISO oo buuxisa heerarka wax soo saarka GMP, la shaqaaleysiiyay khubarada isku dhafka daroogada ee gudaha iyo dibadda oo leh khibrad qani ah si ay u hagaan R&D ee shirkadda.

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Faa'iidooyinka Isbeddelka Caafimaadka

TECHNOL OGY FAA'IIDOOYINKA
●Cadaadiska Sare ee Katalytic Hydrogenation.Cadaadiska Sare ee Hydrogenolysis Falcelinta .Falcelinta Cryogenic (<-78%C)
●Aromatic Heterocyclic Synthesis
● Falcelinta dib u habeynta
●Go'aanka Chiral
●Heck, Suzuki,Negishi,Sonogashira .Falcelinta Gignard

JIN DUN R&D

Qalabka

Shaybaadhkayagu waxa uu leeyahay qalab tijaabo ah oo kala duwan, sida: NMR (Bruker 400M),HPLC,chiral-HPLC,LC-MS,LC-MS/MS (API 4000),IR,UV,GC,GC-MS, Chromatography, Mikrowave Synthesizer, Parallel Synthesizer, Kalorimitirka Iskaanka Kala Duwan (DSC), Microscope Electron...

Kooxda R&D

Jindun Medical waxay leedahay koox shaqaale R&D ah oo xirfad leh, waxayna shaqaaleysiisaa khubaro badan oo gudaha iyo dibedda ah oo ku takhasusay isku-darka daroogada si ay u hagaan R&D, taasoo ka dhigaysa isku-dhafkayaga mid sax ah oo hufan.

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Dacwad- Wadaag

Waxaan caawinay dhowr shirkadood oo dawooyinka gudaha ugu sarreeya, sidaHansoh, Hengrui iyo HEC Pharm.Halkan waxaan ku tusi doonaa qayb iyaga ka mid ah.

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Kiiska Koowaad ee Customization:

Cas No.: 110351-94-5

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Cabashada Labaad:

Cas No.: 144848-24-8

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Kiiska Saddexaad ee Habaynta:

Cas No.: 200636-54-0

Habka iskaashiga

1.Habbee Dhexdhexaadiyeyaasha Cusub ama API-yada.Si la mid ah wadaagista kiisaska kore, macaamiishu waxay leeyihiin dalabaadka Dhexdhexaadiyeyaasha gaarka ah ama API-yada, mana ka heli karaan badeecadaha loo baahan yahay suuqa, ka dib waxaan ku caawin karnaa si aan u habeyno.

2.Habraaca Hagaajinta Alaabta Hore.Kooxdayadu waxay gacan ka geysan doontaa in ay wanaajiso oo ay hagaajiso wax soo saarka noocaas ah oo dariiqa falcelinta ee duugoobay, qiimaha wax soo saarku uu sarreeyo, waxtarkeeduna uu yar yahay.Waxaan ku siin karnaa dukumeenti buuxa oo wareejinta tignoolajiyada iyo hagaajinta habka, ka caawinta macaamiisha wax soo saar hufan.

Laga soo bilaabo bartilmaameedyada daroogada ilaa INDs, JIN DUN Medical ayaa ku siinaysaXalka R&D shaqsiyeysan ee hal-joojin ah.

JIN DUN Medical waxay ku adkaysanaysaa abuurista koox riyooyin leh, samaynta alaab sharaf leh, taxadar leh, adag, iyo u bixista dhammaan si ay u noqoto lammaane la aamini karo iyo saaxiibka macaamiisha!


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